| 发明名称 |
NAPHTHYRIDINE DERIVATIVE MONOHYDRATE AND METHOD FOR PRODUCING THE SAME |
| 摘要 |
Disclosed is 1-(2-(4-((2,3-dihydro(1,4)dioxino(2,3-c)pyridin-7-ylmethyl)amino)piperidin-1-yl)ethyl)-7-fluoro-1,5-naphthyridin-2(1H)-one monohydrate, which has strong antibacterial activity. The compound is highly safe and useful as an original drug for pharmaceutical preparations. Also disclosed is a method which is useful for producing 1-(2-(4-((2,3-dihydro(1,4)dioxino(2,3-c)pyridin-7-ylmethyl)amino)piperidin-1-yl)ethyl)-7-fluoro-1,5-naphthyridin-2(1H)-one monohydrate.
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| 申请公布号 |
EP2221309(A1) |
申请公布日期 |
2010.08.25 |
| 申请号 |
EP20080855286 |
申请日期 |
2008.11.25 |
| 申请人 |
TOYAMA CHEMICAL CO., LTD.;TAISHO PHARMACEUTICAL CO., LTD. |
发明人 |
KIYOTO, TARO;TAKEBAYASHI, MASAHIRO;BABA, YASUTAKA;SYOJI, MUNEO;NOGUCHI, TOSHIYA;USHIYAMA, FUMIHITO;URABE, HIROKI;HORIKIRI, HIROMASA |
| 分类号 |
C07D519/00;A61K31/4545;A61P31/04;C07D309/40;C07D491/04;C07D491/056 |
主分类号 |
C07D519/00 |
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