发明名称 METHOD FOR PREPARING 1-(3-(2-(1-BENZOTHIOPHENE-5-YL)ETHOXY)PROPYL)AZETIDINE-3-OL OR ITS SALTS
摘要 FIELD: medicine, pharmaceutics. ^ SUBSTANCE: invention refers to a method for preparing 1-(3-(2-(1-benzothiophene-5-yl)ethoxy)propyl)azetidine-3-ol or its salts which involves the use as a parent compound, (phenylthio)acetic acid derivative or its salts presented by general formula: where X1 represents halogen atom, and is applicable as a safe method of volume production of 1-(3-(2-(1-benzothiophene-5-yl)ethoxy)propyl)azetidine-3-ol or its salts effective as an agent in disorders of the central nervous system and peripheral nervous system. ^ EFFECT: there is provided high yield, safety for human body, low environment loads. ^ 36 cl, 1 tbl, 33 ex
申请公布号 RU2397169(C2) 申请公布日期 2010.08.20
申请号 RU20070139770 申请日期 2006.03.27
申请人 TOJAMA KEMIKAL KO., LTD. 发明人 SAITOKH AKIKHITO;SUZUKI JOSIAKI;JONEZAVA KENDZI;KAVAMURA MITSUKHIDE;KUSANAGI TAKAKHIKO;NAKAI TAKASI
分类号 C07D333/54;C07D409/12 主分类号 C07D333/54
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