发明名称 AROMATIC DERIVATIVE AS HIV ASPARTYL PROTEASE INHIBITOR
摘要 PROBLEM TO BE SOLVED: To provide a new kind of compounds, and derivatives thereof permissible as pharmaceuticals. SOLUTION: There are provided HIV aspartyl protease inhibitors of the formula (I) and, when the compound of formula (I) contains an amino group, pharmaceutically acceptable ammonium salts thereof, (wherein n is 3 or 4; R<SB>1</SB>may be, for example, iso-butyl; X and Y are same or different, and may be, for example, NH<SB>2</SB>and F; and R<SB>2</SB>and R<SB>3</SB>are as specifically defined herein). COPYRIGHT: (C)2010,JPO&INPIT
申请公布号 JP2010180224(A) 申请公布日期 2010.08.19
申请号 JP20100068414 申请日期 2010.03.24
申请人 AMBRILIA BIOPHARMA INC 发明人 STRANIX BRENT RICHARD;LAVALLEE JEAN-FRANCOIS;LEBERRE NICOLAS;PERRON VALERIE
分类号 C07C311/18;A61K31/145;A61K31/341;A61K31/40;A61K31/4164;A61K31/44;A61K31/4406;A61K31/455;A61K31/4965;A61K31/5375;A61K31/5377;A61P31/18;A61P43/00;C07C311/40;C07C311/41;C07D207/34;C07D213/74;C07D213/78;C07D213/81;C07D233/90;C07D237/24;C07D241/24;C07D295/20;C07D295/215;C07D307/24;C07D317/62 主分类号 C07C311/18
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