发明名称 |
DIAZEPINEDIONE DERIVATIVE |
摘要 |
<p>A diazepinedione derivative represented by general formula (I) or a pharmacologically acceptable salt thereof is used as a P2X4 receptor antagonist. (In the formula, R1 represents a hydrogen atom, a C1-8 alkyl, etc.; R2 and R3 each represents a hydrogen atom, a C1-8 alkyl, a halogen atom, etc.; R4 and R5 each represents a hydrogen atom, a C1-8 alkyl, etc.; and W represents a tetrazole residue, etc.)</p> |
申请公布号 |
WO2010093061(A1) |
申请公布日期 |
2010.08.19 |
申请号 |
WO2010JP52571 |
申请日期 |
2010.02.15 |
申请人 |
NIPPON CHEMIPHAR CO., LTD.;SAKUMA, SHOGO;TAKAHASHI, TOSHIHIRO;USHIODA, MASATOSHI;IMAI, TOSHIYASU;INOUE, KAZUHIDE |
发明人 |
SAKUMA, SHOGO;TAKAHASHI, TOSHIHIRO;USHIODA, MASATOSHI;IMAI, TOSHIYASU;INOUE, KAZUHIDE |
分类号 |
C07D403/10;A61K31/5513;A61P25/04;A61P43/00;C07D413/10;C07D417/10 |
主分类号 |
C07D403/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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