发明名称 AN IMPROVED PROCESS FOR THE PREPARATION OF PALIPERIDONE
摘要 <p>The invention relates to an improved process for the preparation of Pal?peridone in high yield and purity. The purity of Paliperidone is ~99.7 % by HPLC, wherein total impurity is less than about 0.3 % and each individual impurity is less than about 0.1 %. The invention also relates to provide the alcohol-water co-solvent for the purification of Paliperidone.</p>
申请公布号 WO2010089643(A1) 申请公布日期 2010.08.12
申请号 WO2010IB00178 申请日期 2010.02.01
申请人 CADILA PHARMACEUTICALS LTD.;SODAGAR, KEVAL, RAMESHCHANDRA;MALIK, VINEET;JAIN, SUDHIR, HUKAMCHAND;PARIKH, SANJAY, NATVARLAL;SHARMA, ARUN, OMPRAKASH;BAPAT, UDAY, RAJARAM;MODI, INDRAVADAN, AMBALAL 发明人 SODAGAR, KEVAL, RAMESHCHANDRA;MALIK, VINEET;JAIN, SUDHIR, HUKAMCHAND;PARIKH, SANJAY, NATVARLAL;SHARMA, ARUN, OMPRAKASH;BAPAT, UDAY, RAJARAM;MODI, INDRAVADAN, AMBALAL
分类号 A01N43/90 主分类号 A01N43/90
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