发明名称 PROCESS FOR PREPARING OLOPATADINE AND/OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF
摘要 <p>The present invention relates to a process for the preparation of olopatadine and, more particularly, to an improved method of synthesizing olopatadine which comprises reacting a dibenz[b,e]oxepin-1 1-one derivative of formula (III) and a suitable reagent under Witting condition.</p>
申请公布号 WO2010089268(A2) 申请公布日期 2010.08.12
申请号 WO2010EP51148 申请日期 2010.02.01
申请人 ZACH SYSTEM S.P.A.;GUIDI, ALBERTO;CHIARELLO, FILIPPO;ORRU', GIANMAURO;VERZINI, MASSIMO;COTARCA, LIVIUS;KIZIRIAN, JEAN-CLAUDE;TREPAT GUIXER, ELISENDA;MARQUILLAS OLONDRIZ, FRANCISCO 发明人 GUIDI, ALBERTO;CHIARELLO, FILIPPO;ORRU', GIANMAURO;VERZINI, MASSIMO;COTARCA, LIVIUS;KIZIRIAN, JEAN-CLAUDE;TREPAT GUIXER, ELISENDA;MARQUILLAS OLONDRIZ, FRANCISCO
分类号 C07D313/12 主分类号 C07D313/12
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