发明名称 |
XINAFOATE SALT OF N4- (2,2-DIFLUORO-4H-BENZO [1,4] OXAZIN-3-ONE) - 6-YL] - 5-FLUORO-N2 - [3-(METHYLAMINOCARBONYLMETHYLENEOXY) PHENYL] 2,4-PYRIMIDINEDIAMINE |
摘要 |
<p>The present invention relates to the xinafoate salt of N4-[(2,2-difluoro-4H-benzo[1,4]oxazin-3-one)-6-yl]-5-fluoro-N2-[3-(methylaminocarbonylmethyleneoxy)phenyl]-2,4-pyrimidinediamine. This compound is a suitable drug substance and is useful in the treatment of conditions including asthma.</p> |
申请公布号 |
EP2215087(A2) |
申请公布日期 |
2010.08.11 |
申请号 |
EP20080806983 |
申请日期 |
2008.08.27 |
申请人 |
PFIZER LIMITED |
发明人 |
TAYLOR, STEFAN, COLIN, JOHN |
分类号 |
C07D413/12;A61K31/538;A61P11/06 |
主分类号 |
C07D413/12 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|