发明名称 XINAFOATE SALT OF N4- (2,2-DIFLUORO-4H-BENZO [1,4] OXAZIN-3-ONE) - 6-YL] - 5-FLUORO-N2 - [3-(METHYLAMINOCARBONYLMETHYLENEOXY) PHENYL] 2,4-PYRIMIDINEDIAMINE
摘要 <p>The present invention relates to the xinafoate salt of N4-[(2,2-difluoro-4H-benzo[1,4]oxazin-3-one)-6-yl]-5-fluoro-N2-[3-(methylaminocarbonylmethyleneoxy)phenyl]-2,4-pyrimidinediamine. This compound is a suitable drug substance and is useful in the treatment of conditions including asthma.</p>
申请公布号 EP2215087(A2) 申请公布日期 2010.08.11
申请号 EP20080806983 申请日期 2008.08.27
申请人 PFIZER LIMITED 发明人 TAYLOR, STEFAN, COLIN, JOHN
分类号 C07D413/12;A61K31/538;A61P11/06 主分类号 C07D413/12
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