发明名称 |
2-(2-OXOINDOLINE-3-YLIDENE)METHYL-5-(2-HYDROXY-3-MORPHOLIN-4-YL -PROPYL)-6,7-DIHYDRO -1H- PYRROL[3,2-C]PYRIDINE-4(5H)-ONE COMPOUNDS AND USE AS PROTEIN KINASE INHIBITORS |
摘要 |
Pyrrolo[3,2-c]pyridine-4-one-2-indolinone compounds, especially 2-(2-oxoindoline-3-ylidene)methyl-5-(2-hydroxy-3-morpholin-4-yl-propyl)-6,7-dihyd ro-1H-pyrrol[3,2-c]pyridine-4(5H)-one compounds. Their preparation and pharmaceutical composition, and pharmaceutical use as protein kinase inhibitors. |
申请公布号 |
EP2179998(A4) |
申请公布日期 |
2010.07.28 |
申请号 |
EP20080783579 |
申请日期 |
2008.07.29 |
申请人 |
JIANGSU HENGRUI MEDICINE CO., LTD.;SHANGHAI HENGRUI PHARMACEUTICAL CO. LTD. |
发明人 |
TANG, PENG CHO;YANG, JIALIANG;SU, YIDONG;ZHAO, FUQIANG |
分类号 |
C07D417/04;A61K31/437;A61P33/00;C07D209/04;C07D209/30 |
主分类号 |
C07D417/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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