发明名称 THIENO-(1,3)-OXAZIN-4-ONES WITH LIPASE INHIBITING ACTIVITY
摘要 PROBLEM TO BE SOLVED: To provide a compound for treating obesity or obesity-related disorders. SOLUTION: The compound of formula (I) (wherein A is an optionally substituted thienyl moiety; Y is O, S or NR<SP>2</SP>; R<SP>1</SP>is a branched or unbranched alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, aryl, arylalkyl, reduced arylalkyl, arylalkenyl, heteroaryl, heteroarylalkyl, heteroarylalkenyl, reduced aryl, reduced heteroaryl, reduced heteroarylalkyl or a substituted derivative of any of the above groups; and R<SP>2</SP>is hydrogen or a group as defined for R<SP>1</SP>) or a pharmaceutically acceptable salt, ester, amide or prodrug thereof is described. COPYRIGHT: (C)2010,JPO&INPIT
申请公布号 JP2010159260(A) 申请公布日期 2010.07.22
申请号 JP20100019160 申请日期 2010.01.29
申请人 NORGINE BV 发明人 HODSON HAROLD FRANCIS;DUNK CHRISTOPHER ROBERT;PALMER RICHARD MICHAEL JOHN;MITCHELL DALE ROBERT;BIRAULT VERONIQUE;HUNT RUSSELL GEORGE
分类号 A23L1/30;C07D498/04;A23L3/3544;A61K8/49;A61K31/4365;A61K31/535;A61K31/5365;A61P1/00;A61P3/04;A61P3/06;A61P3/10;A61P9/00;A61P9/12;A61P25/00;A61P43/00;A61Q19/10;C07D498/14;C11D3/28;C11D3/48;C12N9/99 主分类号 A23L1/30
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