Described herein are somatostatin analogs that are receptor antagonists of the somatostatin receptor, including SSTR2-selective antagonists. Related compounds, kits and methods, including antagonists complexed with or conjugated to radioactive nuclides and uses thereof. The antagonists of the invention are useful in diagnosing and treating neoplastic and non-neoplastic mammalian diseases.
申请公布号
WO2009129311(A3)
申请公布日期
2010.07.22
申请号
WO2009US40672
申请日期
2009.04.15
申请人
SALK INSTITUTE FOR BIOLOGICAL STUDIES;UNIVERSITAT BERN;UNIVERSITY HOSPITAL BASEL;RIVIER, JEAN, E. F.;ERCHEGYI, JUDIT;REUBI, JEAN, CLAUDE;MAECKE, HELMUT, R.
发明人
RIVIER, JEAN, E. F.;ERCHEGYI, JUDIT;REUBI, JEAN, CLAUDE;MAECKE, HELMUT, R.