发明名称 |
PYRROLOPYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS MEDICAMENTS |
摘要 |
The invention is directed to certain novel compounds. Specifically, the invention is directed to compounds according to formula (I): and salts thereof. The compounds of the invention are inhibitors of kinase activity, in particular IKK2 activity.
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申请公布号 |
US2010179139(A1) |
申请公布日期 |
2010.07.15 |
申请号 |
US20080602619 |
申请日期 |
2008.05.29 |
申请人 |
BAMBOROUGH PAUL;BARKER MICHAEL DAVID;CAMPOS SEBASTIEN ANDRE;COUSINS RICHARD PETER CHARLES;FAULDER PAUL;HOBBS HEATHER;HOLMES DUNCAN STUART;JOHNSTON MICHAEL JOHN;LIDDLE JOHN;PAYNE JEREMY JOHN;PRITCHARD JOHN MARTIN;WHITWORTH CAROLINE |
发明人 |
BAMBOROUGH PAUL;BARKER MICHAEL DAVID;CAMPOS SEBASTIEN ANDRE;COUSINS RICHARD PETER CHARLES;FAULDER PAUL;HOBBS HEATHER;HOLMES DUNCAN STUART;JOHNSTON MICHAEL JOHN;LIDDLE JOHN;PAYNE JEREMY JOHN;PRITCHARD JOHN MARTIN;WHITWORTH CAROLINE |
分类号 |
A61K31/437;A61K31/506;A61K31/541;A61P3/10;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P19/10;A61P25/00;A61P25/28;A61P29/00;A61P31/18;A61P35/00;C07D471/04 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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