发明名称 PYRROLOPYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS MEDICAMENTS
摘要 The invention is directed to certain novel compounds. Specifically, the invention is directed to compounds according to formula (I): and salts thereof. The compounds of the invention are inhibitors of kinase activity, in particular IKK2 activity.
申请公布号 US2010179139(A1) 申请公布日期 2010.07.15
申请号 US20080602619 申请日期 2008.05.29
申请人 BAMBOROUGH PAUL;BARKER MICHAEL DAVID;CAMPOS SEBASTIEN ANDRE;COUSINS RICHARD PETER CHARLES;FAULDER PAUL;HOBBS HEATHER;HOLMES DUNCAN STUART;JOHNSTON MICHAEL JOHN;LIDDLE JOHN;PAYNE JEREMY JOHN;PRITCHARD JOHN MARTIN;WHITWORTH CAROLINE 发明人 BAMBOROUGH PAUL;BARKER MICHAEL DAVID;CAMPOS SEBASTIEN ANDRE;COUSINS RICHARD PETER CHARLES;FAULDER PAUL;HOBBS HEATHER;HOLMES DUNCAN STUART;JOHNSTON MICHAEL JOHN;LIDDLE JOHN;PAYNE JEREMY JOHN;PRITCHARD JOHN MARTIN;WHITWORTH CAROLINE
分类号 A61K31/437;A61K31/506;A61K31/541;A61P3/10;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P19/10;A61P25/00;A61P25/28;A61P29/00;A61P31/18;A61P35/00;C07D471/04 主分类号 A61K31/437
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