发明名称 |
METHOD OF PREPARING (+)-1,4-DIHYDRO-7-[(3S,4S)-3METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID |
摘要 |
Methods of preparing (+)-1, 4-dihydro-7-[(3S,45)-3-methoxy-4-(methylamino)-1 - pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid are disclosed. Also provided are pharmaceutical compositions comprising (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid, and methods of treatment using such compositions. |
申请公布号 |
WO2010078294(A1) |
申请公布日期 |
2010.07.08 |
申请号 |
WO2009US69645 |
申请日期 |
2009.12.29 |
申请人 |
SUNESIS PHARMACEUTICAL, INC.;SUDHAKAR, ANANTHA;SUBRAMANI, TAMILARASAN;RAHUMAN, MOHAMED SHEIK MOHAMED MUJEEBUR;SUBBIAH, RAMAR |
发明人 |
SUDHAKAR, ANANTHA;SUBRAMANI, TAMILARASAN;RAHUMAN, MOHAMED SHEIK MOHAMED MUJEEBUR;SUBBIAH, RAMAR |
分类号 |
C07D471/04;A61K31/4375;A61P35/00;C07D207/14 |
主分类号 |
C07D471/04 |
代理机构 |
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