发明名称 METHOD OF PREPARING (+)-1,4-DIHYDRO-7-[(3S,4S)-3METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID
摘要 Methods of preparing (+)-1, 4-dihydro-7-[(3S,45)-3-methoxy-4-(methylamino)-1 - pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid are disclosed. Also provided are pharmaceutical compositions comprising (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid, and methods of treatment using such compositions.
申请公布号 WO2010078294(A1) 申请公布日期 2010.07.08
申请号 WO2009US69645 申请日期 2009.12.29
申请人 SUNESIS PHARMACEUTICAL, INC.;SUDHAKAR, ANANTHA;SUBRAMANI, TAMILARASAN;RAHUMAN, MOHAMED SHEIK MOHAMED MUJEEBUR;SUBBIAH, RAMAR 发明人 SUDHAKAR, ANANTHA;SUBRAMANI, TAMILARASAN;RAHUMAN, MOHAMED SHEIK MOHAMED MUJEEBUR;SUBBIAH, RAMAR
分类号 C07D471/04;A61K31/4375;A61P35/00;C07D207/14 主分类号 C07D471/04
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