发明名称 |
PROCESS FOR THE PREPARATION OF A MACROCYCLE. |
摘要 |
<p>The present invention relates to a new process for the preparation of macrocyclic HCV protease inhibitor compounds of the formula (VII) wherein R1 is an amino protecting group and X is halogen by way of a ring closing metathesis approach.</p> |
申请公布号 |
MX2010006659(A) |
申请公布日期 |
2010.07.05 |
申请号 |
MX20100006659 |
申请日期 |
2008.12.11 |
申请人 |
F. HOFFMANN-LA ROCHE AG. |
发明人 |
MICHELANGELO SCALONE.;KURT PUENTENER.;STEFAN HILDBRAND |
分类号 |
C07D403/12;C07D487/04 |
主分类号 |
C07D403/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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