发明名称 EG5 INHIBITOR
摘要 <p>Provided is a novel Eg5 inhibitor which contains, as an active ingredient, a nitrogen-containing heteropolycyclic compound such as a carbazole derivative or a carboline derivative.  The novel Eg5 inhibitor contains, as an active ingredient, a nitrogen-containing heteropolycyclic compound represented by general formula (I) or a pharmacologically acceptable salt thereof.  In general formula (I), the linkages a-b and c-d are each a single or double bond; Q1 to Q4 are each a nitrogen atom or -C(X)=; X and Y1 to Y4 are each a hydrogen atom, an alkyl group, an aralky group, an aryl group, a heterocyclic group, a hydroxyl group, an alkoxy group, a carboxyl group, a halogen atom, or the like; and Z is a hydrogen atom, an alkyl group, or the like.</p>
申请公布号 WO2010073719(A1) 申请公布日期 2010.07.01
申请号 WO2009JP07298 申请日期 2009.12.25
申请人 KYOTO UNIVERSITY;PHARMA IP GENERAL INCORPORATED ASSOCIATION;FUJII, NOBUTAKA;OGAWA, OSAMU;NISHIYAMA, HIROYUKI;OHNO, HIROAKI;OISHI, SHINYA;WATANABE, TOSHIAKI;TAKEUCHI, TOMOKI;ASAI, AKIRA;SAWADA, JUNICHI 发明人 FUJII, NOBUTAKA;OGAWA, OSAMU;NISHIYAMA, HIROYUKI;OHNO, HIROAKI;OISHI, SHINYA;WATANABE, TOSHIAKI;TAKEUCHI, TOMOKI;ASAI, AKIRA;SAWADA, JUNICHI
分类号 C07D209/86;C07D471/04;A61K31/403;A61K31/437;A61K31/4745;A61P35/00;A61P37/02;A61P37/06;A61P43/00;C07D209/88 主分类号 C07D209/86
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