摘要 |
<p>Provided is a novel Eg5 inhibitor which contains, as an active ingredient, a nitrogen-containing heteropolycyclic compound such as a carbazole derivative or a carboline derivative. The novel Eg5 inhibitor contains, as an active ingredient, a nitrogen-containing heteropolycyclic compound represented by general formula (I) or a pharmacologically acceptable salt thereof. In general formula (I), the linkages a-b and c-d are each a single or double bond; Q1 to Q4 are each a nitrogen atom or -C(X)=; X and Y1 to Y4 are each a hydrogen atom, an alkyl group, an aralky group, an aryl group, a heterocyclic group, a hydroxyl group, an alkoxy group, a carboxyl group, a halogen atom, or the like; and Z is a hydrogen atom, an alkyl group, or the like.</p> |
申请人 |
KYOTO UNIVERSITY;PHARMA IP GENERAL INCORPORATED ASSOCIATION;FUJII, NOBUTAKA;OGAWA, OSAMU;NISHIYAMA, HIROYUKI;OHNO, HIROAKI;OISHI, SHINYA;WATANABE, TOSHIAKI;TAKEUCHI, TOMOKI;ASAI, AKIRA;SAWADA, JUNICHI |
发明人 |
FUJII, NOBUTAKA;OGAWA, OSAMU;NISHIYAMA, HIROYUKI;OHNO, HIROAKI;OISHI, SHINYA;WATANABE, TOSHIAKI;TAKEUCHI, TOMOKI;ASAI, AKIRA;SAWADA, JUNICHI |