发明名称 NOVEL INTERMEDIATE AND PROCESS FOR PREPARING ENTECAVIR USING SAME
摘要 The present invention relates to a novel, high-yield and low-cost method for preparing entecavir, [1-S-(1a,3a,4,ß]-2-amino-1,9-dihydro-9-[4-hydroxy-3-(hydroxymethyl)-2-methylenecyclopentyl]-6H-purin-6-one, an antiviral agent, and novel intermediates used therein.
申请公布号 WO2010074534(A2) 申请公布日期 2010.07.01
申请号 WO2009KR07786 申请日期 2009.12.24
申请人 HANMI PHARM. CO., LTD.;LEE, JAEHEON;PARK, GHA-SEUNG;KIM, JIN HEE;LEE, JI EUN;PARK, CHUL HYUN;CHOI, TAE JIN;PARK, EUN-JU;KIM, CHEOL KYUNG;LIM, EUN JUNG;CHANG, YOUNG-KIL;LEE, GWAN SUN 发明人 LEE, JAEHEON;PARK, GHA-SEUNG;KIM, JIN HEE;LEE, JI EUN;PARK, CHUL HYUN;CHOI, TAE JIN;PARK, EUN-JU;KIM, CHEOL KYUNG;LIM, EUN JUNG;CHANG, YOUNG-KIL;LEE, GWAN SUN
分类号 C07D473/18 主分类号 C07D473/18
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