| 发明名称 |
2,3-DIHYDROIMINOISOINDOLE DERIVATIVE |
| 摘要 |
<p>A compound represented by the following general formula (1), or a salt thereof has serine protease inhibiting activity, and particularly excellent inhibiting activity against clotting factor VIIa. This compound or a salt thereof is useful as therapeutic and/or prophylactic agents for diseases associated with thrombus formation.
[wherein R 1 represents hydrogen, R 2 represents optionally substituted phenyl, etc., R 3 represents optionally substituted C6-10 aryl, etc.]</p> |
| 申请公布号 |
EP2202231(A1) |
申请公布日期 |
2010.06.30 |
| 申请号 |
EP20080832347 |
申请日期 |
2008.09.19 |
| 申请人 |
EISAI R&D MANAGEMENT CO., LTD. |
发明人 |
CLARK, RICHARD;TAKEMURA, ATSUSHI;WATANABE, NOBUHISA;ASANO, OSAMU;NAGAKURA, TADASHI;TABATA, KIMIYO |
| 分类号 |
C07D401/12;A61K31/4196;A61K31/422;A61K31/427;A61K31/4439;A61K31/506;A61P11/00;A61P7/02;A61P9/10;A61P9/14;A61P35/00;A61P43/00;C07D209/44;C07D401/14;C07D405/14;C07D409/14;C07D413/14;C07D417/14 |
主分类号 |
C07D401/12 |
| 代理机构 |
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