发明名称 |
HALOGENIERTE PYRAZOLOÄ1,5-AÜPYRIMIDINE, VERFAHREN, ANWENDUNGEN ALS GABA-A-REZEPTORLIGAND, ZUSAMMENSETZUNGEN UND ZWISCHENPRODUKTE |
摘要 |
The invention provides novel halogenated pyrazolo[1,5-a]pyrimidines of formula (I) wherein R, R 1 , X and Y have different meanings, and pharmaceutically acceptable salts thereof. Compounds of formula (I) are useful for treating or preventing anxiety, epilepsy and sleep disorders including insomnia, and for inducing sedation-hypnosis, anesthesia, sleep and muscle relaxation. The invention also provides synthetic procedures for preparing said compounds and certain intermediates, as well as intermediates themselves. |
申请公布号 |
DE602006014272(D1) |
申请公布日期 |
2010.06.24 |
申请号 |
DE20066014272T |
申请日期 |
2006.06.15 |
申请人 |
FERRER INTERNACIONAL S.A. |
发明人 |
ANGLADA, LUIS;PALOMER, ALBERT;GUGLIETTA, ANTONIO |
分类号 |
C07D487/04;A61K31/519;A61P25/08;A61P25/20;A61P25/22;C07C211/21 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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