发明名称 SPIRO (FURO [3, 2-C] PYRIDINE-3-3' -INDOL) -2' (1'H)-ONE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SODIUM-CHANNEL MEDIATED DISEASES, SUCH AS PAIN
摘要 This invention is directed to methods of using spiro-oxindole compounds of formula (I): wherein j, k, m, Q, X, R1, R2a, R2b, R2c, R2d and R3 are as defined herein, as a stereoisomer, enantiomer, tautomer thereof or mixtures thereof; or a pharmaceutically acceptable salt, N-oxide, solvate or prodrug thereof, for the treatment and/or prevention of sodium channel-mediated diseases or conditions, such as pain.
申请公布号 US2010160362(A1) 申请公布日期 2010.06.24
申请号 US20070445270 申请日期 2007.10.12
申请人 XENON PHARMACEUTICALS INC. 发明人 CADIEUX JEAN-JACQUES;CHOWDHURY SULTAN;FU JIANMIN;KAMBOJ RAJENDER;HSIEH TOM;JIA QI;LIU SHIFENG;SUN JIANYU
分类号 A61K31/438;C07D491/20 主分类号 A61K31/438
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