发明名称 PROCESSES FOR PREPARING 5,7 DIAMINOPYRAZOLO[1,5-a] PYRIMIDINE COMPOUNDS
摘要 Processes for the preparation of certain 5,7-diaminopyrazolo[1,5-a]pyrimidine compounds comprising the reaction of a primary or secondary amine and a protected 5-halo-7-aminopyrazolo[1,5-a]pyrimidine compound in solvent system comprising water and one or more organic solvents, optionally in the presence of an exogenous base.
申请公布号 WO2010068838(A2) 申请公布日期 2010.06.17
申请号 WO2009US67627 申请日期 2009.12.11
申请人 EMORY UNIVERSITY;IMPERIAL COLLEGE OF SCIENCE AND TECHNOLOGY;LIOTTA, DENNIS, C.;SNYDER, JAMES, P.;JOGALEKAR, ASHUTOSH, S.;BARRETT, ANTHONY, G.M.;FUCHTER, MATTHEW, JOHN;COOK, MATTHEW, J.;KROLL, SEBASTIAN, H.B. 发明人 LIOTTA, DENNIS, C.;SNYDER, JAMES, P.;JOGALEKAR, ASHUTOSH, S.;BARRETT, ANTHONY, G.M.;FUCHTER, MATTHEW, JOHN;COOK, MATTHEW, J.;KROLL, SEBASTIAN, H.B.
分类号 C07D487/04;C07D487/02 主分类号 C07D487/04
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