发明名称 NONSTEROIDAL LIGAND FOR GLUCOCORTICOID RECEPTOR, COMPOSITION THEREOF, AND USE THEREOF
摘要 PROBLEM TO BE SOLVED: To provide a method for treating or preventing obesity, diabetes, anxiety, depression, neurodegeneration, or inflammatory diseases. SOLUTION: There are provided a nonsteroidal ligand for glucocorticoid receptors, a method for producing a nonsteroidal ligand for glucocorticoid receptors, and methods for using a nonsteroidal ligand for glucocorticoid receptors and nonsteroidal ligand compositions. These are effective against diseases associated with the binding between a glucocorticoid and a glucocorticoid receptor, for examples, obesity, diabetes, depression, neurodegeneration, or inflammatory diseases. COPYRIGHT: (C)2010,JPO&INPIT
申请公布号 JP2010132672(A) 申请公布日期 2010.06.17
申请号 JP20100006117 申请日期 2010.01.14
申请人 REGENTS OF THE UNIV OF CALIFORNIA 发明人 SCANLAN THOMAS S;SHAH NILESH
分类号 C07D231/54;A61K31/415;A61K31/416;A61K31/4162;A61K31/42;A61K31/423;A61K31/425;A61P3/04;A61P3/10;A61P5/44;A61P5/46;A61P25/00;A61P25/22;A61P25/24;A61P25/28;A61P29/00;A61P43/00;C07D275/06;C07D317/72;C07D327/10;C07D339/06;C07D403/06;C07D409/06;C07D487/04 主分类号 C07D231/54
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