发明名称 IMIDAZOPYRIDAZINES FOR USE AS PROTEIN KINASE INHIBITORS
摘要 There is provided compounds of formula (I): wherein Z, M, R1, X, R3, R4 and R5 have meanings given in the description, an pharmaceutically-acceptable esters, amides, solvates or salts thereof, which compounds are useful in the treatment of diseases in which inhibition of a protein kinase (e.g. a PIM family kinase or PI3-K) is desired and/or required, an particularly in the treatment of cancer.
申请公布号 WO2009060197(A8) 申请公布日期 2010.06.17
申请号 WO2008GB03744 申请日期 2008.11.10
申请人 CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO);PEVARELLO, PAOLO;GARCIA COLLAZO, ANA MARIA;RODRIGUEZ HERGUETA, ANTONIO;SALUSTE, CARL-GUSTAF PIERRE;RAMOS LIMA, FRANCISCO JAVIER;GONZALEZ CANTALAPIEDRA, ESTHER;OYARZABAL SANTAMARINA, JULEN 发明人 PEVARELLO, PAOLO;GARCIA COLLAZO, ANA MARIA;RODRIGUEZ HERGUETA, ANTONIO;SALUSTE, CARL-GUSTAF PIERRE;RAMOS LIMA, FRANCISCO JAVIER;GONZALEZ CANTALAPIEDRA, ESTHER;OYARZABAL SANTAMARINA, JULEN
分类号 C07D487/04;A61K31/519;A61P35/00 主分类号 C07D487/04
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