发明名称 POLY-HETEROARYL DERIVATIVES FOR THE TREATMENT OF CANCER
摘要 <p>The present invention relates to Penta- hexa-, hepta-, octa-, nona- and, deca-heteroaryl derivatives, comprising a combination of heterocycle 1 (Het-1)a and/or heterocycie 2 (Het-2)b and/ or heterocycle 3 (Het-3)c and/or heterocycle 4 (Het-4)d of formulae I, II, III and IV respectively, the N-oxides, the pharmaceutically acceptable addition salts. The compounds claimed are suitable for the treatment of cancer.</p>
申请公布号 WO2010049915(A8) 申请公布日期 2010.06.17
申请号 WO2009IB54856 申请日期 2009.11.02
申请人 INSTITUT CURIE;CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS);INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM);MUSEUM NATIONAL D'HISTOIRE NATURELLE (MNHN);NGUYEN, CHI-HUNG;ROUCHON DAGOIS, MYRIAM;GUEDIN-BEAUREPAIRE, AURORE;MONCHAUD, DAVID;TEULADE-FICHOU, MARIE-PAULE;RIOU, JEAN-FRANCOIS;MERGNY, JEAN-LOUIS;GRIERSON, DAVID 发明人 NGUYEN, CHI-HUNG;ROUCHON DAGOIS, MYRIAM;GUEDIN-BEAUREPAIRE, AURORE;MONCHAUD, DAVID;TEULADE-FICHOU, MARIE-PAULE;RIOU, JEAN-FRANCOIS;MERGNY, JEAN-LOUIS;GRIERSON, DAVID
分类号 C07D413/14;A61K31/4439;A61K31/444;A61K31/496;A61P35/00 主分类号 C07D413/14
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