发明名称 ONE-POT PRODUCTION PROCESS FOR CINNAMIDE DERIVATIVE
摘要 <p>A compound represented by the formula (1) below or a pharmaceutically acceptable salt thereof is able to be produced in one pot by reacting a compound represented by the formula (2) below with 3-methoxy-4-(4-methyl-1H-imidazol-1-yl)benzaldehyde in the presence of a base and, if necessary, removing a protecting group. (In the formula (2), R 1 represents a 4-fluorophenyl group or the like; Q represents -CH(CH 3 )-or the like; and n represents 1 or the like.) (In the formula (1), R represents a 4-fluorophenyl group or the like; Q and n are as defined above.)</p>
申请公布号 IL202098(D0) 申请公布日期 2010.06.16
申请号 IL20090202098 申请日期 2009.11.12
申请人 EISAI R& D MANAGEMENT CO., LTD. 发明人
分类号 C07D 主分类号 C07D
代理机构 代理人
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