SYNTHESIS AND NOVEL SALT FORMS OF (R)-5-((E)-2-(PYRROLIDIN-3-YLVINYL)PYRIMIDINE
摘要
The present invention relates to the stereospecific synthesis of (R)-5-((E)-2-pyrrolidin-3-ylvinyl)pyrimidine, its salt forms, and novel polymorphic forms of these salts.
申请公布号
CA2742366(A1)
申请公布日期
2010.06.10
申请号
CA20092742366
申请日期
2009.11.30
申请人
TARGACEPT, INC.
发明人
AKIREDDY, SRINIVISA RAO;BHATTI, BALWINDER SINGH;CUTHBERTSON, TIMOTHY J.;DULL, GARY MAURICE;MILLER, CRAIG HARRISON;MITCHENER, JOSEPH PIKE, JR.;MUNOZ, JULIO A.;OTTEN, PIETER ALBERT