发明名称 SYNTHESIS AND NOVEL SALT FORMS OF (R)-5-((E)-2-(PYRROLIDIN-3-YLVINYL)PYRIMIDINE
摘要 The present invention relates to the stereospecific synthesis of (R)-5-((E)-2-pyrrolidin-3-ylvinyl)pyrimidine, its salt forms, and novel polymorphic forms of these salts.
申请公布号 CA2742366(A1) 申请公布日期 2010.06.10
申请号 CA20092742366 申请日期 2009.11.30
申请人 TARGACEPT, INC. 发明人 AKIREDDY, SRINIVISA RAO;BHATTI, BALWINDER SINGH;CUTHBERTSON, TIMOTHY J.;DULL, GARY MAURICE;MILLER, CRAIG HARRISON;MITCHENER, JOSEPH PIKE, JR.;MUNOZ, JULIO A.;OTTEN, PIETER ALBERT
分类号 C07D403/06;A61K31/505;A61P25/00 主分类号 C07D403/06
代理机构 代理人
主权项
地址