发明名称 SYNTHESIS AND NOVEL SALT FORMS OF (R)-5-((E)-2-(PYRROLIDIN-3-YLVINYL)PYRIMIDINE
摘要 The present invention relates to the stereospecific synthesis of (R)-5-((E)-2-pyrrolidin-3-ylvinyl)pyrimidine, its salt forms, and novel polymorphic forms of these salts.
申请公布号 WO2010065443(A1) 申请公布日期 2010.06.10
申请号 WO2009US66078 申请日期 2009.11.30
申请人 TARGACEPT, INC.;AKIREDDY, SRINIVISA RAO;BHATTI, BALWINDER, SINGH;CUTHBERTSON, TIMOTHY, J.;DULL, GARY, MAURICE;MILLER, CRAIG, HARRISON;MITCHENER, JR., JOSEPH, PIKE;MUNOZ, JULIO, A.;OTTEN, PIETER, ALBERT 发明人 AKIREDDY, SRINIVISA RAO;BHATTI, BALWINDER, SINGH;CUTHBERTSON, TIMOTHY, J.;DULL, GARY, MAURICE;MILLER, CRAIG, HARRISON;MITCHENER, JR., JOSEPH, PIKE;MUNOZ, JULIO, A.;OTTEN, PIETER, ALBERT
分类号 C07D403/06;A61K31/505;A61P25/00 主分类号 C07D403/06
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