发明名称 |
FUSED HETEROARYL DERIVATIVES |
摘要 |
The present invention provides a pharmaceutical composition which is useful as a phosphatidylinositol 3 kinase (PI3K) inhibitor and an antitumor agent, and it provides a novel bicyclic or tricyclic fused heteroaryl derivative or a salt thereof which possesses an excellent PI3K inhibiting activity and cancer cell growth inhibiting activity.
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申请公布号 |
US2010137585(A1) |
申请公布日期 |
2010.06.03 |
申请号 |
US20100688273 |
申请日期 |
2010.01.15 |
申请人 |
HAYAKAWA MASAHIKO;KAIZAWA HIROYUKI;MORITOMO HIROYUKI;KAWAGUCHI KEN-ICHI;KOIZUMI TOMONOBU;YAMANO MAYUMI;MATSUDA KOYO;OKADA MINORU;OHTA MITSUAKI |
发明人 |
HAYAKAWA MASAHIKO;KAIZAWA HIROYUKI;MORITOMO HIROYUKI;KAWAGUCHI KEN-ICHI;KOIZUMI TOMONOBU;YAMANO MAYUMI;MATSUDA KOYO;OKADA MINORU;OHTA MITSUAKI |
分类号 |
C07D487/04;A61K31/00;A61K31/517;A61K31/519;A61K31/5377;C07D471/04;C07D471/14;C07D491/04;C07D491/048;C07D491/14;C07D495/04;C07D495/14 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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地址 |
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