发明名称 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM
摘要 <p>The present invention relates to compounds defined by formula (I), wherein the groups X, Y, W and R1 to R4 are defined as in claim 1, possessing valuable pharmacological activity. Particularly the compounds are agonists of the 5-HT2C receptor, and thus are suitable for treatment and prevention of diseases which can be influenced by inhibition of this receptor, such as metabolic and CNS-related disorders.</p>
申请公布号 WO2010060952(A1) 申请公布日期 2010.06.03
申请号 WO2009EP65883 申请日期 2009.11.26
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH;MUELLER, STEPHAN-GEORG;BROWN, CHRISTOPER, JOHN;HEIFETZ, ALEXANDER;NOSSE, BERND;PRESTLE, JUERGEN;PREVOST, NATACHA;RUDOLF, KLAUS;SCHEUERER, STEFAN;SCHINDLER, MARCUS;STENKAMP, DIRK;THOMAS, LEO;TYE, HEATHER 发明人 MUELLER, STEPHAN-GEORG;BROWN, CHRISTOPER, JOHN;HEIFETZ, ALEXANDER;NOSSE, BERND;PRESTLE, JUERGEN;PREVOST, NATACHA;RUDOLF, KLAUS;SCHEUERER, STEFAN;SCHINDLER, MARCUS;STENKAMP, DIRK;THOMAS, LEO;TYE, HEATHER
分类号 C07D487/14;A61K31/519;A61P3/00;A61P25/00 主分类号 C07D487/14
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