发明名称 7-PYRIDINYL- OR PHENYL- SUBSTITUTED TRIAZOLO [1, 5 -A] PYRIDINES AS PI3K INHIBITORS
摘要 <p>The invention relates to compounds of formula (I), wherein X, X1, R and R1 to R4 have the meaning as cited in the description and the claims. Said compounds are useful as protein kinase inhibitors, especially inhibitors of PI3K, for the treatment or prophylaxis of immunological, inflammatory, autoimmune, or allergic disorders. The invention also relates to pharmaceutical compositions including said compounds, the preparation of such compounds as well as the production of and use as medicaments.</p>
申请公布号 WO2010057877(A1) 申请公布日期 2010.05.27
申请号 WO2009EP65292 申请日期 2009.11.17
申请人 CELLZOME LIMITED;RAMSDEN, NIGEL;BELL, KATHRYN;TAYLOR, JESS;SUNOSE, MIHIRO;MIDDLEMISS, DAVID;ELLARD, KATIE 发明人 RAMSDEN, NIGEL;BELL, KATHRYN;TAYLOR, JESS;SUNOSE, MIHIRO;MIDDLEMISS, DAVID;ELLARD, KATIE
分类号 A61K31/437;C07D471/04;A61P3/00;A61P29/00;A61P35/00;A61P37/08 主分类号 A61K31/437
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