摘要 |
Nitrilopyrimidin derivatives of general formula (I):, (I)whereinB is CR, where Ris hydrogen, -C-C-alkyl, -C-Calkenyl, -C-Calkynyl, -C-C-cycloalkyl, -C-Ccarboxy, - COO-C-alkyl, aryl, heteroaryl, each is optionally substituted by halogen, - O-C-C-alkyl, -S-C-alkyl, -C-C-cycloalkyl, CN, NO, -NH, -NH(C-C-alkyl), -N(C-C-alkyl), -NHCO(C-C-alkyl), phenyl;D is CRor N, where Ris hydrogen, -C-Calkyl, -C-Calkenyl, -C-Calkynyl, -C-C-cycloalkyl, -CO-C-alkyl, CN, aryl, heteroaryl, each is optionally substituted by halogen, O-C-C-alkyl, -S-C-C-alkyl, -C-C-cycloalkyl, CN, NO, -NH, -NH(C-C-alkyl), -N(C-C-alkyl), -NHCO(C-C-alkyl), phenyl. |