发明名称 GAMMA SECRETASE MODULATORS
摘要 <p>In its many embodiments, the present invention provides a novel class of heterocyclic compounds of the formula: as modulators of gamma secretase, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more diseases associated with the central nervous system using such compounds or pharmaceutical compositions.</p>
申请公布号 WO2010056722(A1) 申请公布日期 2010.05.20
申请号 WO2009US63993 申请日期 2009.11.11
申请人 SCHERING CORPORATION;ZHU, ZHAONING;GREENLEE, WILLIAM, J.;LI, HONGMEI;VICAREL, MONICA, L.;QIN, JUN;DHONDI, PAWAN, KUMAR;HUANG, XIANHAI;PALANI, ANANDAN;LIU, XIAOXIANG;SUN, ZHONG-YUE;JOSIEN, HUBERT B.;XU, RUO;COLE, DAVID, JAMES;BURNETT, DUANE, A.;BENNETT, CHAD, E.;MCCRACKEN, TROY, M.;MACCOSS, MALCOLM 发明人 ZHU, ZHAONING;GREENLEE, WILLIAM, J.;LI, HONGMEI;VICAREL, MONICA, L.;QIN, JUN;DHONDI, PAWAN, KUMAR;HUANG, XIANHAI;PALANI, ANANDAN;LIU, XIAOXIANG;SUN, ZHONG-YUE;JOSIEN, HUBERT B.;XU, RUO;COLE, DAVID, JAMES;BURNETT, DUANE, A.;BENNETT, CHAD, E.;MCCRACKEN, TROY, M.;MACCOSS, MALCOLM
分类号 C07D409/14;A61K31/5395;A61K31/553;A61P25/28;C07D413/10;C07D498/04;C07D498/14;C07D498/20 主分类号 C07D409/14
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