发明名称 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS
摘要 The present invention relates to a compounds of formula I wherein R1, R2, R3, R4, R5, and n are as defined herein and to a pharmaceutically active salt, a racemic mixture, an enantiomer, an optical isomer or a tautomeric form thereof. The present compounds are high potential NK-3 receptor antagonists for the treatment of depression, pain, psychosis, Parkinson's disease, schizophrenia, anxiety and attention deficit hyperactivity disorder (ADHD).
申请公布号 US2010125078(A1) 申请公布日期 2010.05.20
申请号 US20090614474 申请日期 2009.11.09
申请人 KNUST HENNER;LIMBERG ANJA;NETTEKOVEN MATTHIAS;RATNI HASANE;RIEMER CLAUS;VIFIAN WALTER 发明人 KNUST HENNER;LIMBERG ANJA;NETTEKOVEN MATTHIAS;RATNI HASANE;RIEMER CLAUS;VIFIAN WALTER
分类号 A61K31/498;A61K31/517;A61P25/18;C07D401/14;C07D403/04 主分类号 A61K31/498
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