发明名称 GERING HYGROSKOPISCHE ARIPIPRAZOL-SUBSTANZ (KRISTAL E) UND HERSTELLUNGSVERFAHREN
摘要 The present invention provides low-hygroscopic forms of aripiprazole and processes for the preparation thereof which will not convert to a hydrate or lose their original solubility even when a medicinal preparation containing the aripiprazole anhydride crystals is stored for an extended period.
申请公布号 AT467416(T) 申请公布日期 2010.05.15
申请号 AT20080000360T 申请日期 2002.09.25
申请人 OTSUKA PHARMACEUTICAL CO., LTD. 发明人 BANDO, TAKUJI;AOKI, SATOSHI;KAWASAKI, JUNICHI;ISHIGAMI, MAKOTO;TANIGUCHI, YOUICHI;YABUUCHI, TSUYOSHI;FUJIMOTO, KIYOSHI;NISHIOKA, YOSHIHIRO;KOBAYASHI, NORIYUKI;FUJIMURA, TSUTOMU;TAKAHASHI, MASANORI;ABE, KAORU;NAKAGAWA, TOMONORI;SHINHAMA, KOICHI;UTSUMI, NAOTO;TOMINAGA, MICHIAKI;OI, YOSHIHIRO;YAMADA, SHOHEI;TOMIKAWA, KENJI
分类号 A61K31/496;C07D215/22;A61K;A61K9/14;A61K9/16;A61K9/20;A61K31/4704;A61K31/501;A61P;A61P1/08;A61P3/04;A61P15/10;A61P25/00;A61P25/04;A61P25/16;A61P25/18;A61P25/22;A61P25/28;A61P25/32;B01D9/02;C07D;C07D215/227 主分类号 A61K31/496
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