发明名称 |
PROCESS TO PREPARE NEW SUBSITUTED 1H-BENZO[d]IMIDAZOL-2(3H)-ONES, NEW INTERMEDIATES AND THEIR USE AS BACE 1 INHIBITORS |
摘要 |
The invention relates to a new process leading to new substituted 1H-benzo[d]imidazol-2(3H)-ones of formula III and III′, to pharmaceutical compositions comprising them and to their use as therapeutic agents, particularly as BACE 1 inhibitors in the treatment of Alzheimer disease.
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申请公布号 |
US2010120880(A1) |
申请公布日期 |
2010.05.13 |
申请号 |
US20080329739 |
申请日期 |
2008.12.08 |
申请人 |
UNIVERSITE PAUL CEZANNE-AIX MARSEILLE III |
发明人 |
ROUSSEL CHRISTIAN;ANDREOLI FEDERICO;VANTHUYNE NICOLAS DANIEL PIERRE |
分类号 |
A61K31/4184;A61P25/28;C07D235/04 |
主分类号 |
A61K31/4184 |
代理机构 |
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