发明名称 Piperidinylamino-thieno[2,3-D] Pyrimidine Compounds
摘要 The invention relates to 5-HT receptor modulators, particularly 5-HT2B antagonists. Novel piperidinylamino-thieno[2,3-d]pyrimidine compounds represented by Formula I, II and III, and uses thereof for treating conditions including pulmonary arterial hypertension, congestive heart failure, and hypertension.
申请公布号 US2010113485(A1) 申请公布日期 2010.05.06
申请号 US20090609470 申请日期 2009.10.30
申请人 DHANOA DALE S;BECKER OREN;NOIMAN SILVIA;ALLA SEKAR REDDY;CHERUKU SRINIVASA RAO;MELE NDEZ ROSA E;SHARADENDU ANURAG;CHEN DONGLI;MARANTZ YAEL;SHACHAM SHARON;HEIFETZ ALEXANDER;INBAL BOAZ;KESAVAN VENKITASAMY;BAR-HAIM SHAY 发明人 DHANOA DALE S.;BECKER OREN;NOIMAN SILVIA;ALLA SEKAR REDDY;CHERUKU SRINIVASA RAO;MELE'NDEZ ROSA E.;SHARADENDU ANURAG;CHEN DONGLI;MARANTZ YAEL;SHACHAM SHARON;HEIFETZ ALEXANDER;INBAL BOAZ;KESAVAN VENKITASAMY;BAR-HAIM SHAY
分类号 A61K31/519;A61P1/00;A61P5/00;A61P5/08;A61P9/00;A61P9/12;A61P11/00;A61P11/06;A61P15/00;A61P15/10;A61P19/00;A61P25/00;A61P25/06;A61P25/22;A61P25/24;A61P25/28;A61P29/00;A61P35/00;C07D495/04;C07D498/02 主分类号 A61K31/519
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