发明名称 |
Piperidinylamino-thieno[2,3-D] Pyrimidine Compounds |
摘要 |
The invention relates to 5-HT receptor modulators, particularly 5-HT2B antagonists. Novel piperidinylamino-thieno[2,3-d]pyrimidine compounds represented by Formula I, II and III, and uses thereof for treating conditions including pulmonary arterial hypertension, congestive heart failure, and hypertension.
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申请公布号 |
US2010113485(A1) |
申请公布日期 |
2010.05.06 |
申请号 |
US20090609470 |
申请日期 |
2009.10.30 |
申请人 |
DHANOA DALE S;BECKER OREN;NOIMAN SILVIA;ALLA SEKAR REDDY;CHERUKU SRINIVASA RAO;MELE NDEZ ROSA E;SHARADENDU ANURAG;CHEN DONGLI;MARANTZ YAEL;SHACHAM SHARON;HEIFETZ ALEXANDER;INBAL BOAZ;KESAVAN VENKITASAMY;BAR-HAIM SHAY |
发明人 |
DHANOA DALE S.;BECKER OREN;NOIMAN SILVIA;ALLA SEKAR REDDY;CHERUKU SRINIVASA RAO;MELE'NDEZ ROSA E.;SHARADENDU ANURAG;CHEN DONGLI;MARANTZ YAEL;SHACHAM SHARON;HEIFETZ ALEXANDER;INBAL BOAZ;KESAVAN VENKITASAMY;BAR-HAIM SHAY |
分类号 |
A61K31/519;A61P1/00;A61P5/00;A61P5/08;A61P9/00;A61P9/12;A61P11/00;A61P11/06;A61P15/00;A61P15/10;A61P19/00;A61P25/00;A61P25/06;A61P25/22;A61P25/24;A61P25/28;A61P29/00;A61P35/00;C07D495/04;C07D498/02 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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