发明名称 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS
摘要 Heterocyclic compounds that bind chemokine receptors and inhibit the binding of their natural ligands are disclosed. The invention compounds are protective against infection by HIV and exert effects characteristic of antagonists to the CXCR4 receptor.
申请公布号 US2010105915(A1) 申请公布日期 2010.04.29
申请号 US20090612488 申请日期 2009.11.04
申请人 BRIDGER GARY J;SKERLJ RENATO;KALLER AI;HARWIG CURTIS;BOGUCKI DAVID;WILSON TREVOR R;CRAWFORD JASON;MCEACHERN ERNEST J;ATSMA BEM;NAN SIQIAO;ZHOU YUANXI;SCHOLS DOMINIQUE 发明人 BRIDGER GARY J.;SKERLJ RENATO;KALLER AI;HARWIG CURTIS;BOGUCKI DAVID;WILSON TREVOR R.;CRAWFORD JASON;MCEACHERN ERNEST J.;ATSMA BEM;NAN SIQIAO;ZHOU YUANXI;SCHOLS DOMINIQUE
分类号 C07D401/02;A61K31/4402;A61K31/4439;A61K31/444;A61K31/46;A61K31/4709;A61K31/4725;A61K31/4985;A61K31/5377;A61K45/06;A61P1/04;A61P3/10;A61P5/14;A61P11/00;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P17/12;A61P19/02;A61P21/00;A61P21/04;A61P29/00;A61P31/18;A61P35/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D213/36;C07D213/38;C07D215/40;C07D239/42;C07D401/12;C07D401/14;C07D405/14;C07D409/14;C07D413/14;C07D417/14;C07D451/04;C07D471/04;C07D487/04 主分类号 C07D401/02
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