发明名称 NOVEL CRYSTALS AND PROCESS OF MAKING 5-({[2-AMINO-3-(4-CARBAMOYL-2,6-DIMETHYL-PHENYL)-PROPIONYL]-[1-(4-PHENYL-1H-IMIDAZOL-2-YL)-ETHYL]-AMINO}-METHYL)-2-METHOXY-BENZOIC ACID
摘要 The present invention relates to a novel crystals of 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid and methods of making the zwitterion of 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid.
申请公布号 KR20100043210(A) 申请公布日期 2010.04.28
申请号 KR20107002535 申请日期 2008.07.07
申请人 JANSSEN PHARMACEUTICA N. V 发明人 ANZALONE LUIGI;VILLANI FRANK J.;TELEHA CHRISTOPHER ALLAN;FEIBUSH PENINA;FEGELY BARRY
分类号 C07D233/64;A61K31/4164;A61P1/00 主分类号 C07D233/64
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