发明名称 |
HETEROCYCLYL AND CYCLOALKYL SUBSTITUTED THIENO[2,3-D]PYRIMIDINE AND THEIR USE AS ADENOSINE A2A RECEPTOR ANTAGONISTS |
摘要 |
This invention relates to a novel thieno[2,3-d]pyrimidine, Z, and its therapeutic and prophylactic uses, wherein X, R1 and R2 are defined in the specification. Disorders treatedand/or prevented include Parkinson's Disease.Formula (I).
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申请公布号 |
CA2740525(A1) |
申请公布日期 |
2010.04.22 |
申请号 |
CA20092740525 |
申请日期 |
2009.09.29 |
申请人 |
JANSSEN PHARMACEUTICA NV |
发明人 |
BARBAY, J. KENT;LEONARD, KRISTI;CHAKRAVARTY, DEVRAJ;SHOOK, BRIAN CHRISTOPHER;WANG, AIHUA |
分类号 |
C07D495/04;A61K31/519;A61P25/00 |
主分类号 |
C07D495/04 |
代理机构 |
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