发明名称 |
Arylamidine derivative, salt thereof, and antifungal containing these |
摘要 |
An arylamidine derivative represented by the general formula (wherein R1 represents optionally protected or substituted amidino; and R2 and R3 are the same or different and each represents hydrogen or halogeno) or a salt of the derivative. The derivative and salt have potent activity against fungi including ones having tolerance to azole type drugs and further have high safety and excellent properties in a repeated dose toxicity test. They are hence useful as an excellent antifungal.
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申请公布号 |
US7700623(B2) |
申请公布日期 |
2010.04.20 |
申请号 |
US20050631399 |
申请日期 |
2005.06.28 |
申请人 |
TOYAMA CHEMICAL CO., LTD. |
发明人 |
HAYASHI KAZUYA;KUNITANI KAZUTO;UEHARA SAYURI;MORITA TEIICHI |
分类号 |
A61K31/445;A01N43/42;A61K31/435;C07D211/20 |
主分类号 |
A61K31/445 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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