发明名称 |
5-PHENYLTHIAZOLE DERIVATIVES AND USE AS PI3 KINASE INHIBITORS |
摘要 |
Compounds of formula I in free or salt form, wherein R1, R2, R3, R4 and R5 have the meanings as indicated in the specification, are useful for treating diseases mediated by phosphatidylinositol 3-kinase. Pharmaceutical compositions that contain the compounds and processes for preparing the compounds are also described.
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申请公布号 |
US2010093690(A1) |
申请公布日期 |
2010.04.15 |
申请号 |
US20090640479 |
申请日期 |
2009.12.17 |
申请人 |
BRUCE IAN;FINAN PETER;LEBLANC CATHERINE;MCCARTHY CLIVE;WHITEHEAD LEWIS;PRESS NICOLA;BLOOMFIELD GRAHAM CHARLES;HAYLER JUDY;KIRMAN LOUISE;OZA MRINALINI SACHIN;SHUKLA LENA |
发明人 |
BRUCE IAN;FINAN PETER;LEBLANC CATHERINE;MCCARTHY CLIVE;WHITEHEAD LEWIS;PRESS NICOLA;BLOOMFIELD GRAHAM CHARLES;HAYLER JUDY;KIRMAN LOUISE;OZA MRINALINI SACHIN;SHUKLA LENA |
分类号 |
A61K31/397;C07D277/20;A61K31/426;A61K31/427;A61K31/4436;A61K31/4439;A61K31/496;A61K31/5377;A61P1/04;A61P3/04;A61P3/10;A61P7/08;A61P9/00;A61P9/10;A61P11/00;A61P17/06;A61P19/02;A61P29/00;A61P31/04;A61P35/00;A61P37/06;A61P37/08;A61P43/00;C07D277/42;C07D277/44;C07D277/46;C07D277/48;C07D413/14;C07D417/02;C07D417/04;C07D417/12 |
主分类号 |
A61K31/397 |
代理机构 |
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