发明名称 PERIPHERAL OPIOID RECEPTOR ANTAGONISTS AND USES THEREOF
摘要 The present invention provides a compound of formula I: wherein X-, R1, and R2 are as defined herein, and compositions thereof. The compounds are peripheral opioid receptors.
申请公布号 WO2010039851(A1) 申请公布日期 2010.04.08
申请号 WO2009US59058 申请日期 2009.09.30
申请人 WYETH LLC;BAZHINA, NATALIYA;DONATO, GEORGE, JOSEPH;FABIAN, STEVEN, R.;LOKHNAUTH, JOHN;MEGATI, SREENIVASULU;MELUCCI, CHARLES;OFSLAGER, CHRISTIAN;PATEL, NIKETA;RADEBAUGH, GALEN;SHAH, SYED, M.;SZELIGA, JAN;ZHANG, HUYI;ZHU, TIANMIN 发明人 BAZHINA, NATALIYA;DONATO, GEORGE, JOSEPH;FABIAN, STEVEN, R.;LOKHNAUTH, JOHN;MEGATI, SREENIVASULU;MELUCCI, CHARLES;OFSLAGER, CHRISTIAN;PATEL, NIKETA;RADEBAUGH, GALEN;SHAH, SYED, M.;SZELIGA, JAN;ZHANG, HUYI;ZHU, TIANMIN
分类号 C07D471/08;A61K31/485;A61P1/10;C07D489/08 主分类号 C07D471/08
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