发明名称 |
2-[1H-Benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides as kinase inhibitors |
摘要 |
2-[1H-benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and their salts are kinase inhibitors, useful in the treatment of cancer.
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申请公布号 |
US2010081653(A1) |
申请公布日期 |
2010.04.01 |
申请号 |
US20090567060 |
申请日期 |
2009.09.25 |
申请人 |
TELIK, INC. |
发明人 |
AURRECOECHEA NATALIA;BEROZA PAUL P.;DAMODARAN KOMATH V.;PONTIUS KAREN Y.;ROBINSON LOUISE;SIMON REYNA J.;VU TRUONG;WEBER KEVIN T. |
分类号 |
A61K31/506;A61K31/496;A61K31/5377;A61K31/541;C07D401/14;C07D403/06;C07D403/14;C07D413/14;C07D417/06;C07D417/14 |
主分类号 |
A61K31/506 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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