发明名称 2-[1H-Benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides as kinase inhibitors
摘要 2-[1H-benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and their salts are kinase inhibitors, useful in the treatment of cancer.
申请公布号 US2010081653(A1) 申请公布日期 2010.04.01
申请号 US20090567060 申请日期 2009.09.25
申请人 TELIK, INC. 发明人 AURRECOECHEA NATALIA;BEROZA PAUL P.;DAMODARAN KOMATH V.;PONTIUS KAREN Y.;ROBINSON LOUISE;SIMON REYNA J.;VU TRUONG;WEBER KEVIN T.
分类号 A61K31/506;A61K31/496;A61K31/5377;A61K31/541;C07D401/14;C07D403/06;C07D403/14;C07D413/14;C07D417/06;C07D417/14 主分类号 A61K31/506
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