发明名称 SULFUR CONTAINING PYRAZOLE-HETEROCYCLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS
摘要 A novel sulfur containing heteroaryl-pyrazole compound of formula (I) or a pharmaceutically acceptable salt thereof is effective as a cannabinoid CB1 receptor inverse agonist or antagonist, which is useful for preventing or treating obesity and obesity-related metabolic disorders. The prevention also provide a method for preparing same, a pharmaceutical composition containing same, and a method for preventing or treating obesity and obesity-related metabolic disorders.
申请公布号 WO2010035915(A1) 申请公布日期 2010.04.01
申请号 WO2008KR05689 申请日期 2008.09.25
申请人 GREEN CROSS CORPORATION;LEE, JINHWA;SEO, HEE JEONG;KIM, MIN-AH;KIM, JEONGMIN;LEE, SUNG-HAN;JUNG, MYUNG EUN;KIM, MI-SOON 发明人 LEE, JINHWA;SEO, HEE JEONG;KIM, MIN-AH;KIM, JEONGMIN;LEE, SUNG-HAN;JUNG, MYUNG EUN;KIM, MI-SOON
分类号 A61K31/4164;C07D265/30;A61K51/04;C07D233/54 主分类号 A61K31/4164
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