2-[1H-BENZIMIDAZOL-2(3H)-YLIDENE]-2-(PYRIMIDIN-2-YL)ACETAMIDES AND 2-[BENZOTHIAZOL-2(3H)-YLIDENE]-2-(PYRIMIDIN-2-YL)ACETAMIDES AS KINASE INHIBITORS
摘要
2-[1H-benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and their salts are kinase inhibitors, useful in the treatment of cancer. Formula I
申请公布号
CA2734472(A1)
申请公布日期
2010.04.01
申请号
CA20092734472
申请日期
2009.09.25
申请人
TELIK, INC.
发明人
AURRECOECHEA, NATALIA;BEROZA, PAUL P.;DAMODARAN, KOMATH V.;PONTIUS, KAREN Y.;ROBINSON, LOUISE;SIMON, REYNA J.;VU, TRUONG;WEBER, KEVIN T.