发明名称 POLYMORPHS OF 5--6-CHLORO-1,3-DIHYDRO-2H-INDOL-2-ONE HYDROBROMIDE AND PROCESSES FOR PREPARATION THEREOF
摘要 The present invention provides pharmaceutically applicable compounds and polymorphs belonging to the ziprasidone hydrobromide compound group with antipsychotic effect. The present invention provides hydrobromide polymorphs of 5-{-2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]-ethyl}-6-chloro-1,3-dihydro-2H-indol-2-one, ziprasidone of Formula (I) having neuroleptic activity.
申请公布号 US2010081668(A1) 申请公布日期 2010.04.01
申请号 US20070516094 申请日期 2007.11.23
申请人 NEU JOZSEF;DEMETER ADAM;VARGA ZOLTAN;HAVASI BALAZS;GARADNAY SANDOR;HEGEDUES BELA 发明人 NEU JOZSEF;DEMETER ADAM;VARGA ZOLTAN;HAVASI BALAZS;GARADNAY SANDOR;HEGEDUES BELA
分类号 A61K31/496;A61P25/00;C07D417/14 主分类号 A61K31/496
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