发明名称 |
POLYMORPHS OF 5--6-CHLORO-1,3-DIHYDRO-2H-INDOL-2-ONE HYDROBROMIDE AND PROCESSES FOR PREPARATION THEREOF |
摘要 |
The present invention provides pharmaceutically applicable compounds and polymorphs belonging to the ziprasidone hydrobromide compound group with antipsychotic effect. The present invention provides hydrobromide polymorphs of 5-{-2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]-ethyl}-6-chloro-1,3-dihydro-2H-indol-2-one, ziprasidone of Formula (I) having neuroleptic activity.
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申请公布号 |
US2010081668(A1) |
申请公布日期 |
2010.04.01 |
申请号 |
US20070516094 |
申请日期 |
2007.11.23 |
申请人 |
NEU JOZSEF;DEMETER ADAM;VARGA ZOLTAN;HAVASI BALAZS;GARADNAY SANDOR;HEGEDUES BELA |
发明人 |
NEU JOZSEF;DEMETER ADAM;VARGA ZOLTAN;HAVASI BALAZS;GARADNAY SANDOR;HEGEDUES BELA |
分类号 |
A61K31/496;A61P25/00;C07D417/14 |
主分类号 |
A61K31/496 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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