发明名称 |
Substituted benzimidazoles and imidazo-[4,5]-pyridines |
摘要 |
2-Aryl substituted benzimidazoles and imidazo[4,5]pyridines are disclosed as inhibitors of Cds1 and useful as adjuvants to chemotherapy or radiation therapy in the treatment of cancer.
|
申请公布号 |
US7687639(B2) |
申请公布日期 |
2010.03.30 |
申请号 |
US20060478802 |
申请日期 |
2006.06.30 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
AMERIKS MICHAEL K.;ARIENTI KRISTEN L.;AXE FRANK U.;BREITENBUCHER J. GUY |
分类号 |
C07D235/18;A01N43/52;A61K31/4184;A61K31/454;A61K31/4745;A61P43/00;C07D401/10;C07D401/12;C07D403/12;C07D405/10;C07D405/12;C07D409/12;C07D471/02 |
主分类号 |
C07D235/18 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|