发明名称 LARGE CYCLIC SERINE PROTEASE INHIBITOR OF HEPATITIS C
摘要 <p><P>PROBLEM TO BE SOLVED: To provide a large cyclic compound, and to provide a method for using the large cyclic compound. <P>SOLUTION: A pharmaceutical composition is provided. The composition comprises a compound, e.g., tert-butyl(2R,6S,13aS,14aR,16aS,Z)-2-(3-(benzo[d]thiazol-2-yl)quinoxalin-2-yloxy)-14a-(cyclopropylsulfonylcarbamoyl)-5,16-dioxo-1,2,3,5,6,7,8,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diaza cyclopentadecin-6-yl carbamate or its pharmaceutically permissible salt, ester or prodrug, in combination with a pharmaceutically permissible carrier or excipient. <P>COPYRIGHT: (C)2010,JPO&INPIT</p>
申请公布号 JP2010065035(A) 申请公布日期 2010.03.25
申请号 JP20090208935 申请日期 2009.09.10
申请人 ABBOTT LAB;ENANTA PHARMACEUTICALS INC 发明人 KU YIYIN;MCDANIEL KEITH F;CHEN HUI-JU;SHANLEY JASON P;KEMPF DALE J;GRAMPOVNIK DAVID J;SUN YING;LIU DONG;GAI YONGHUA;OR YAT SUN;WAGAW SABLE H;ENGSTROM KEN;GRIEME TIM
分类号 C07D487/04;A61K31/473;A61K31/498;A61K31/506;A61P31/12;A61P43/00 主分类号 C07D487/04
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