发明名称 |
CRYSTALLINE FORMS OF A 3-PYRROLE SUBSTITUTED 2-INDOLINONE MALATE SALT |
摘要 |
Disclosed are crystalline polymorphic forms of the malic acid salt of (Z)-N-[2- (diethylamino)ethyl]-5-[(5-fluoro-l,2-dihydro-2-oxo-3H-indol-3-yliden)methyl]-2,4- dimethyl-1H-pyrrole-3-carboxamide, sunitinib malate, including crystalline Forms III, IV, V, VI and VII. Also disclosed are processes for preparing crystalline polymorphic forms of sunitinib malate and pharmaceutical compositions comprising sunitinib malate. |
申请公布号 |
WO2010010454(A3) |
申请公布日期 |
2010.03.18 |
申请号 |
WO2009IB06347 |
申请日期 |
2009.07.24 |
申请人 |
MEDICHEM, S.A.;WINTER, STEPHEN, BENEDICT, DAVID;BENITO VELEZ, MONICA |
发明人 |
WINTER, STEPHEN, BENEDICT, DAVID;BENITO VELEZ, MONICA |
分类号 |
C07D403/06;A61K31/404;A61P35/00 |
主分类号 |
C07D403/06 |
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