发明名称 |
A PROCESS FOR PREPARING [1S- [1-ALPHA, 2-ALPHA, 3-BETA (1S*, 2R*) 5-BETA] ] -3- [7- [2- (3, 4-DIF LUOROPHENYL) -CYCLOPROPYLAMINO] - 5- (PROPYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D] PYRIMIDIN-3-YL] -5- (2- HYDROXYETHOXY) CYCLOPENTANE-1, 2-DIOL AND TO ITS INTERMEDIATES |
摘要 |
The present invention is directed to a process for preparing [1S-[1a,2a,3ß(1S*,2R*),5ß]]- 3-[7-[2-(3,4-difluorophenyl)-cyclopropylamino]-5-(propylthio)-3H-1,2,3-triazolo[4,5- d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)cyclopentane-l,2-diol and to intermediates useful in the process.
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申请公布号 |
CA2734454(A1) |
申请公布日期 |
2010.03.18 |
申请号 |
CA20092734454 |
申请日期 |
2009.09.08 |
申请人 |
ASTRAZENECA AB |
发明人 |
AUFDENBLATTEN, RHONY;BOHLIN, MARTIN HANS;HELLSTROEM, HELENA;JOHANSSON, PETER W.;LARSSON, ULF G.;RECKNAGEL, MIKAELA;WEISS, ANDREAS |
分类号 |
C07D487/04;C07D317/44;C07D405/04;C07D405/12 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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地址 |
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