发明名称 |
3-SUBSTITUTED-1H-INDOLE, 3-SUBSTITUTED-1H-PYRROLO[2,3-B]PYRIDINE AND 3-SUBSTITUTED-1H-PYRROLO[3,2-B]PYRIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES |
摘要 |
<p>The invention relates to 3-substituted-1H-indole, 3-substituted-1H-pyrrolo[2,3-b]pyridine, and 3-substituted-1H-pyrrolo[3,2-b]pyridine compounds of the Formula (I): or a pharmaceutically acceptable salt thereof, wherein the constituent variables are as defined herein, compositions comprising the compounds, and methods for making and using the compounds.</p> |
申请公布号 |
WO2010030727(A1) |
申请公布日期 |
2010.03.18 |
申请号 |
WO2009US56443 |
申请日期 |
2009.09.10 |
申请人 |
WYETH LLC;AYRAL-KALOUSTIAN, SEMIRAMIS;MANSOUR, TAREK SUHAYL;TSOU, HWEI-RU;ZHANG, NAN;VENKATESAN, ARANAPAKAM M.;DI, LI;KERNS, EDWARD H. |
发明人 |
AYRAL-KALOUSTIAN, SEMIRAMIS;MANSOUR, TAREK SUHAYL;TSOU, HWEI-RU;ZHANG, NAN;VENKATESAN, ARANAPAKAM M.;DI, LI;KERNS, EDWARD H. |
分类号 |
C07D407/06;A61K31/404;A61P35/00;C07D471/04 |
主分类号 |
C07D407/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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