发明名称 |
NOVEL CRYSTAL FORMS OF 4-(2-AMINOPYRIDIN-4-YL)-3-(4-FLUOROPHENYL)-1-(1,4,5,6-TETRAHYDRO-6-OXOPYRIDAZIN-3-YL)-1H-PYRAZOLE METHANESULFONATE AND METHODS FOR THEIR PREPARATION |
摘要 |
Novel crystal forms of 4-(2-aminopyridin-4-yl)-3-(4- fluorophenyl)-1-(1,4,5,6-tetrahydro-6-oxopyridazin-3-yl)-1H-pyrazole methanesulfonate, which are useful as medicines; and a process for production of same. Two stable polymorphic forms called A-type crystal and B-type crystal; and a process for production by which the polymorphic forms can be each produced as a single polymorphic form.
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申请公布号 |
CA2736554(A1) |
申请公布日期 |
2010.03.18 |
申请号 |
CA20092736554 |
申请日期 |
2009.09.09 |
申请人 |
UBE INDUSTRIES, LTD. |
发明人 |
SHIMIZU, MOTOHISA;SUZUKI, NAOTO;MOTOYAMA, TAKAHIRO;MIYATA, HIROYUKI |
分类号 |
C07D401/14;A61K31/501;A61P19/02;A61P29/00;A61P43/00 |
主分类号 |
C07D401/14 |
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